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CLDN2,CYP3A4,HP,ORM1

Dalam dokumen Supplemental Materials and Methods (Halaman 120-200)

LAP+OC.2- vs LAP+OC.2+

HIBADH 3-hydroxyisobutyrate HIBADH 3-hydroxyisobutyrate dehydrogenase Hist1h1a histone cluster 1, H1a

1.33 CLDN2,CYP3A4,HP,ORM1

SP1 transcriptio

n regulator

Activated 1.33 ABHD2,ACSL1,ALDH3A2,ANKH,ASS1,CBS/CBSL,CEACAM1,CTH,Cyp2d1/Cyp 2d5,EGFR,ESR1,F7,GDF15,GHR,IGF1,IGFBP4,LCAT,PCK1,SGK1

SLC9A3R1 other 1.33 EGFR,SLC34A2

LRPAP1 other 1.33 LRP1,SERPINA3

SAT1 enzyme 1.33 AMY2A,PRKAA2

SPINT1 other 1.33 CLDN2,IGFBP4

ENPP2 3.36 enzyme 1.33 CIDEA,ENPP2

SPARC -5.651 other 1.31 CIDEC,CYP8B1,GPD1,P2RY2,SLC34A2,TSKU

Creb group Activated 1.31 ARG1,CD14,CIDEC,CPT1A,G6PC,GDA,IGF1,ORM1,PCK1,PRKAA2

BRCA1 transcriptio

n regulator

1.31 CYP3A4,EGFR,ENPP2,ESR1,GDF15,MX1,NFE2L2,PERP

LIF cytokine 1.31 CRP,DCAF11,FBP1,IGF1,LBP,SERPINA3,SOCS2,TMEM176A,TMEM176B

Sphk group 1.30 IL33

PLEKHM1 other 1.30 SQSTM1

SMPD3 enzyme 1.30 IGF1

IGF2BP2 -3.166 translation regulator

1.30 LIMS2

APBB2 other 1.30 LRP1

EIF2A translation regulator

1.30 ATF5

TTC7A other 1.30 EGFR

CYP26B1 enzyme 1.30 ATF5

MEX3C other 1.30 IGF1

ADGRG1 g-protein

coupled receptor

1.30 IGF1

MDC1 other 1.30 CLU

SAMHD1 enzyme 1.30 MX1

ZNF385B other 1.30 PERP

ECI1 enzyme 1.30 CYP4A11

MTSS1 other 1.30 EGFR

FBLIM1 other 1.30 EGFR

GFRA1 transmemb

rane receptor

1.30 ACPP

KLHL40 other 1.30 TP53INP1

CD93 other 1.30 CYP27A1

CASP7 peptidase 1.30 CASP4

DAB2IP other 1.30 CLU

EDF1 transcriptio

n regulator

1.30 NR0B2

ABHD5 enzyme 1.30 PDK4

PCBD1 transcriptio

n regulator

1.30 PAH

PTGIS enzyme 1.30 CYP2E1

ASH2L transcriptio

n regulator

1.30 ESR1

TRPC6 ion

channel

1.30 MX1

HNRNPL other 1.30 CEACAM1

MED24 transcriptio

n regulator

1.30 HTRA1

WASHC1 other 1.30 EGFR

DMPK kinase 1.30 FXYD1

GCKR other 1.30 GCK

GCDH enzyme 1.30 ANG

EPHA4 kinase 1.30 IGF1

CIDEA 5.466 other 1.30 XDH

CDO1 20.552 enzyme 1.30 IGF1

CTTN other 1.30 EGFR

PLCD4 enzyme 1.30 EGFR

NDUFS1 enzyme 1.30 GPX1

NOLC1 transcriptio

n regulator

1.30 ORM1

NBN other 1.30 CLU

MAP3K8 kinase 1.27 ACPP,ARG1,ARRDC3,HP,INHBA,SDR42E1,Urah

ADCYAP1 other 1.20 AMACR,ATRN,ENPP2,GCLM,MREG,ORM1,P2RY2,SERPINA3,SERPINF1,UGT2

B28

CDKN2A transcriptio

n regulator

Activated 0.00 Ccl9,CRP,PSMB9,TOB1,TP53INP1

AdH vs LAP+/-, Upstream Regulators, Downregulated in LAP+/-

Upstream Regulator

Expr Fold Change

Molecule Type

Predicted Activation

State

-log(p value)

Target molecules in dataset

TGFB1 growth

factor

Inhibited 21.18 AFP,ANXA2,BGN,BMP2,C1QB,CAV1,Ccl2,CCNA2,CCND2,CCNE1,CD55,CDH5,CX CL10,CXCL2,CXCL3,DAB2,DCN,EDNRB,F2R,FABP5,FCER1G,FLNA,FOS,FXYD6, GSN,GSTA5,GUCY2C,HMOX1,IGF2,IGFBP2,IGFBP7,IL18,IL1A,LGALS3,LIFR,LPL, LYVE1,MCM2,Mcpt1,MFAP4,MKI67,PCNA,PHGDH,PLAGL1,PLEK2,RAMP2,RASG RP3,RBM3,S100A10,S100A11,SERPINH1,SLC25A4,SLC2A1,SLC4A1,SLC7A5,SOCS 3,SPARC,TGFBR3,TIMP1,TIMP3,Tpm4,TSPAN7,TUBA1A,VCAM1,VIM

SP1 transcriptio

n regulator

Inhibited 17.60 ADAMTS1,ADD3,ALAS2,ANK1,CAV1,Ccl2,CCNA2,CCND2,CD55,CDC25B,CXCL1 0,CXCL3,F2R,FLNA,FOS,HBB,HBG2,HDC,HMOX1,IGF2,IL1A,KLF1,LPL,Mt1,NDR G1,PTN,PTTG1,SLC25A4,SLC2A1,SPARC,SPTB,TGFBR3,TIMP1,UGCG,VIM Vegf group Inhibited 15.32 A2M,ADAMTS1,BMP2,CA2,CALCRL,Ccl2,CDC25B,CDH5,CPA3,CXCL10,EMCN,E

MP1,FLNA,GRB10,HDC,HMOX1,IL18,IL1A,KLF1,LYVE1,MCM2,MKI67,PLK1,PMP 22,SKP2,SOCS3,TIMP1,TPX2,UGCG,VCAM1,VIM

MYC transcriptio n regulator

Inhibited 14.75 ADAMTS1,AFP,ALDOA,Bex3,CAV1,CCNA2,CCND2,CCNE1,CD48,CDC25B,CXCL1 0,EMP1,F2R,FABP5,FLNA,FOS,GPC3,H19,HMOX1,IGF2BP1,LDHB,LUM,MCM6,M KI67,Mt1,NDRG1,PCNA,PLK1,PMP22,PSAT1,PTN,RBBP7,S100A10,SERPINH1,SKP 2,SLC2A1,SLC7A5,SPARC,TAGLN2,TIMP1,TSPAN7,VCAM1,VIM

E2F3 transcriptio

n regulator

Inhibited 14.20 CA12,CCNA2,CCNE1,HIST1H2BG,HIST1H4B,IGF2,KIAA0101,LPL,MCM2,MCM4,M CM6,PCNA,PLK1,PTN,PTTG1,SERPINH1,TIMP3,TPX2

HGF growth

factor

Inhibited 13.54 A2M,ADAMTS1,AFP,BMP2,CALCRL,CAV1,Ccl2,CDC25B,CXCL2,EMP1,FLNA,FOS ,GRB10,HMOX1,LYVE1,MCM2,MKI67,PCNA,PLK1,PMP22,PTTG1,SKP2,SOCS3,TA GLN2,TIMP1,TIMP3,TPX2,VCAM1,VIM

TSC2 other Activated 12.78 A2M,ANXA2,Ccl2,CCND2,CXCL10,FOS,GPNMB,GSN,HMOX1,LGALS3,LOC10036 2769,PLP2,S100A11,SLC2A1,UCP2

IKBKB kinase Inhibited 12.56 AFP,BMP2,Ccl2,CCNA2,CDC25B,CXCL10,CXCL2,CXCL3,DCN,FOS,HMOX1,IGFBP 2,IL1A,LIFR,Mt1,OGN,PLK1,SKP2,SOCS3,TIMP3,VCAM1

FGF2 growth

factor

12.41 AFP,BGN,CAV1,CCND2,DCN,EDNRB,FLNA,FOS,GPNMB,IGF2,IGFBP2,LYVE1,M KI67,PCNA,PTTG1,S100A10,SLC2A1,SOCS3,SPARC,TGFBR3,TIMP1,TIMP3,VCAM 1,VIM

TNF cytokine 11.91 A2M,AQP7,ARHGDIB,BGN,BMP2,CA2,CAV1,Ccl2,CCND2,CD55,CDH5,CPA3,CXC L10,CXCL2,CXCL3,DCN,EDNRB,EGLN3,EMCN,EMP1,FABP5,FCER1G,FOS,GSTP1 ,H19,HDC,HMOX1,HPGDS,IGF2,IGFBP2,IL18,IL1A,LGALS3,LIFR,LPL,LYVE1,Mt1, OGN,PDK3,PHGDH,RNASE1,SLC2A1,SOCS3,SPARC,TIMP1,TIMP3,UCP2,UGCG,V CAM1,VIM

EPO cytokine 11.74 ALAS2,ANK1,CA1,CA2,CCND2,FABP5,FOS,HBB,HBG2,IGF2,IL18,KLF1,LCP1,PCN A,Podxl,RHAG,SKP2,SLC4A1,SOCS3,UCP2,UGCG

IL1B cytokine Inhibited 11.58 A2M,ADAMTS1,BGN,BMP2,Ccl2,CD55,CXCL10,CXCL2,CXCL3,DAB2,DCN,EGLN3 ,FABP5,FOS,H19,HMOX1,HPGDS,IL18,IL1A,LCP1,LIFR,Mcpt1,Mt1,RNASE1,S100A 10,SERPINH1,SLC25A4,SLC2A1,SOCS3,SPARC,TIMP1,TIMP3,UGCG,VCAM1,VIM

JUN transcriptio

n regulator

Inhibited 10.93 A2M,AFP,ANXA2,CAV1,Ccl2,CCNA2,CCND2,CXCL10,CXCL3,FOS,GSTA5,GSTP1, HMOX1,IGFBP2,IGFBP7,IL1A,LGALS3,PLAGL1,S100A10,SOCS3,SPARC,TIMP1,V CAM1,VIM

CCL2 cytokine Inhibited 10.77 Ccl2,CXCL10,CXCL3,EGLN3,FOS,HDC,IL18,IL1A,MKI67,PCNA,TIMP1,VCAM1

KITLG growth

factor

Inhibited 10.48 CA2,Ccl2,CCNA2,CCNE1,EDNRB,FABP5,FOS,HMOX1,IL18,IL1A,KLF1,Podxl,RBBP 7,RHAG,SLC4A1,Tpm4,UCP2,UGCG

TP53 transcriptio

n regulator

10.45 A2M,ADD3,AFP,ANXA2,CAV1,Ccl2,CCNA2,CCND2,CCNE1,CDC25B,F2R,FOS,GS N,GSTP1,H19,HDC,Hist1h1b,HMOX1,IGF2,IGFBP2,IGFBP7,IL1A,KIAA0101,LGALS 3,MCM2,MCM4,MCM6,MKI67,NDRG1,PCNA,PHGDH,PLK1,PPIC,PTTG1,RBBP7,R BM3,SERPINH1,SLC2A1,TAGLN2,TIMP3,Tpm4,TPX2,TUBB,VIM

Alpha catenin group Activated 10.43 ADAMTS1,BGN,CXCL10,CXCL2,IGF2,IGFBP2,IGFBP7,LUM,RHOJ,SOCS3,STEAP2, TIMP1,VCAM1,VIM

HIF1A transcriptio Inhibited 10.26 ADAMTS1,AFP,ALDOA,BGN,BMP2,CAV1,Ccl2,CXCL2,CXCL3,EGLN3,FOS,HIF3A,

n regulator HMOX1,IGF2,IGFBP2,IL1A,LIFR,NDRG1,SLC25A37,SLC2A1,SOCS3,VIM

APP other Inhibited 10.03 ALDOA,CA12,Ccl2,CCND2,CCNE1,CDH5,CXCL10,CXCL2,CXCL3,DCN,DPYSL2,F LNA,FOS,GSTP1,H19,HBG2,HMOX1,IGF2,IGF2BP2,IGFBP2,IL18,IL1A,LDB2,LDHB ,LGALS3,Mt1,OGN,PLK1,RELN,SOCS3,TUBA1A,TUBB,VCAM1

IL6 cytokine Inhibited 10.00 A2M,ADAMTS1,AFP,BGN,BMP2,Ccl2,CCNA2,CCNE1,CD48,CXCL10,CXCL2,CXCL 3,DCN,FOS,HMOX1,IGF2,KIAA0101,LIFR,LPL,MKI67,Mt1,Mt1m/Mt2A,PCNA,PTTG 1,SOCS3,STOM,TIMP1,VCAM1,VIM

ADCYAP1 other 9.99 ADD3,Ccl2,CCNA2,CXCL10,CXCL2,CXCL3,EMB,FOS,GPC3,Hmgb2 (includes others),LUM,MCM2,PLAGL1,S100A10,SLC2A1,SOCS3,SPARC,UCP2

P38 MAPK group Inhibited 9.97 ANK1,BGN,BMP2,CAV1,Ccl2,CCND2,CCNE1,CD55,CXCL10,CXCL3,EDNRB,FLNA ,FOS,HMOX1,IL1A,PCNA,SOCS3,TIMP1,TIMP3,TNNI1,VCAM1

Histone h3 group 9.95 ADD3,AFP,ANK1,CAV1,Ccl2,CCNA2,CCND2,CCNE1,CXCL10,ERMAP,FOS,HOXA5 ,IL1A,MCM2,MCM4,Mt1,PCNA,RELN,SOCS3,SPTA1,STOM,Tpm4

NFKBIA transcriptio

n regulator

Inhibited 9.69 A2M,BMP2,Ccl2,CCNA2,CCND2,CDC25B,CXCL10,CXCL2,CXCL3,DCN,FOS,HMO X1,IGF2,IL1A,LIFR,Mt1,OGN,PCNA,SOCS3,TCEAL9,TIMP1,TIMP3,VCAM1

AGT 4.19 growth

factor

Inhibited 9.52 ADD3,BGN,CAV1,Ccl2,CCND2,CCNE1,CXCL10,CXCL2,CXCL3,DAB2,EDNRB,FOS ,GSTA5,GSTP1,HMOX1,IL18,NDRG1,SLC2A1,SOCS3,TIMP1,UCP2,UGCG,VCAM1 INSR kinase Inhibited 9.40 Ccl2,CCND2,DLK1,FOS,GRB10,H19,IFITM2,IGF2,LCP1,LDB2,MCM2,MCM4,NDN,

NDRG1,OGN,PLAGL1,SLC2A1,SOCS3,TNNI1,UCP2,VCAM1

PPARG ligand-

dependent nuclear receptor

9.38 AQP7,CA2,CAV1,Ccl2,CXCL2,CXCL3,DLK1,EGLN3,ELOVL6,FABP5,HMOX1,IGFB P7,LPL,MKI67,NDRG1,PCNA,PPIC,SLC2A1,SOCS3,TUBB,UCP2,VCAM1,VIM

HRAS enzyme 9.34 A2M,AFP,ANXA2,CAV1,Ccl2,CCNA2,CCND2,CCNE1,CXCL10,CXCL2,F2R,FLNA,F OS,GSN,HDC,HMOX1,IFITM2,IGF2,PCNA,PLK1,PPIC,RBBP7,SPARC,TIMP3,Tpm4, VIM

FOS -5.28 transcriptio

n regulator

Inhibited 9.29 A2M,CA2,CCNA2,CCNE1,ELOVL6,EMB,FOS,GSTA5,GSTP1,HMOX1,HPGDS,IL1A, LGALS3,LPL,PLAGL1,PTTG1,RBBP7,S100A10,SOCS3,TIMP1,Tpm4,TUBB,UGCG,V CAM1,VIM

Akt group 9.26 A2M,BMP2,Ccl2,CCND2,CXCL10,FOS,HIF3A,HMOX1,IGF2,IGFBP2,LPL,NDRG1,P CNA,PTN,SKP2,SOCS3,VCAM1

Pdgf (complex) complex 9.22 CAV1,Ccl2,CCND2,CXCL3,FOS,HMOX1,MCM6,PCNA,SPARC,TIMP1,TIMP3,VCA M1

CHUK kinase Inhibited 9.18 BMP2,Ccl2,CXCL10,CXCL2,CXCL3,DCN,FOS,HMOX1,IL1A,LIFR,Mt1,OGN,PCNA, PLK1,SOCS3,VCAM1

OSM cytokine 9.16 A2M,ADAMTS1,AFP,ANXA2,AQP7,ATP2B4,CBX3,Ccl2,CCND2,CXCL10,CXCL2,C XCL3,FOS,GPNMB,HMOX1,IL18,LIFR,PCNA,SOCS3,TIMP1,TIMP3,TPX2,TUBA1A, VCAM1

IL4 cytokine Inhibited 8.97 ANXA2,APOLD1,CA2,CBX3,Ccl2,CCND2,CCNE1,CD55,CXCL10,CXCL2,CXCL3,F2

R,FCER1G,FOS,IL18,IL1A,LGALS2,LGALS3,LIFR,NDRG1,PMP22,S100A10,SLC2A1 ,SOCS3,TFEC,TIMP1,TIMP3,VCAM1,VIM

Ins1 other Inhibited 8.94 AQP7,CCNE1,DLK1,ELOVL6,FOS,GSTP1,IGF2,IGFBP2,LDHB,LIFR,LPL,Mt1,PCNA, SLC2A1,SOCS3,SPARC,TIMP1,TIMP3,VIM

NFkB (complex) complex Inhibited 8.86 A2M,ALDH1B1,BMP2,Ccl2,CCND2,CDC25B,CXCL10,CXCL2,CXCL3,EDNRB,FABP 5,FOS,HIF3A,HMOX1,IGFBP2,IL18,IL1A,PLK1,SLC2A1,SLC7A5,SOCS3,TFEC,TIM P1,VCAM1,VIM

CDKN1A kinase Activated 8.77 CCNA2,CCNE1,CDC25B,CPA3,DTL,KIAA0101,LGALS3,MCM2,MCM4,MCM6,MKI 67,PCNA,PHGDH,PLK1,SKP2,TPX2

SMAD3 transcriptio

n regulator

Inhibited 8.77 BGN,BMP2,Ccl2,CCND2,CCNE1,CDH5,CXCL10,CXCL3,FOS,HMOX1,LUM,PCNA,S LC25A4,TIMP1,TIMP3,VIM

Tgf beta group 8.71 BGN,CCND2,CCNE1,CXCL10,CXCL2,DAB2,DCN,FOS,HMOX1,IL1A,SOCS3,SPAR C,TIMP1,TIMP3,VCAM1,VIM

CTNNB1 transcriptio

n regulator

Inhibited 8.69 AFP,BGN,BMP2,CCNA2,CCND2,CCNE1,Cd52,F2R,FCER1G,FOS,HOXA5,IGF2,IGF2 BP1,IGFBP2,LGALS3,LPL,OGN,PCNA,PLK1,PMP22,Podxl,RCN1,TIMP1,TIMP3,UG CG,VCAM1,VIM

IGF1 21.76 growth

factor

Inhibited 8.69 A2M,BGN,BMP2,Ccl2,CCNA2,CCND2,CCNE1,FOS,HBB,HDC,HMOX1,IGF2,IGFBP2 ,IL18,LPL,MKI67,PCNA,SLC2A1,SOCS3,VCAM1,VIM

MYD88 other Inhibited 8.65 Ccl2,CXCL10,CXCL2,CXCL3,EDNRB,FOS,HDC,HMOX1,IL18,IL1A,MCM2,MKI67,S OCS3,TFEC,TIMP1,VCAM1

ESR2 ligand-

dependent nuclear receptor

8.61 ADAMTS1,ANK1,BMP2,CA12,CA2,CAV1,CCNA2,CLEC1B,EMB,FOS,GSTA5,GSTP 1,LPL,MKI67,NDRG1,PSAT1,RELN,SKP2,SLC25A4,SOCS3,TIMP1

MGEA5 enzyme 8.60 C1QB,CALCRL,CAV1,Ccl2,CD48,CD55,DAB2,FLNA,GSN,HPGDS,IGF2,IGFBP7,IL1 8,PRKAR1B,SOCS3,TGFBR3,TIMP1,TIMP3,TUBA1A,VIM

LIF cytokine 8.44 A2M,AFP,BMP2,Ccl2,CCNA2,CCNE1,CDH5,CXCL10,CXCL2,FOS,LIFR,LPL,SOCS3, TIMP1,TSPAN7

PPARA ligand-

dependent nuclear receptor

8.41 ANXA2,AQP7,C1QB,Ccl2,CCNA2,CCNE1,ELOVL6,FABP5,FOS,GSTP1,HMOX1,IGF BP2,LIFR,LPL,Mcpt1,MKI67,PCNA,PLK1,RBP2,UCP2,VCAM1

TRPV4 ion

channel

Inhibited Ccl2,CXCL10,CXCL2,FOS,SOCS3,TIMP1,VCAM1

CEBPB transcriptio

n regulator

Inhibited Ccl2,CCNA2,CCND2,CCNE1,CDC25B,CXCL2,CXCL3,DAB2,DCN,EMCN,FOS,HBB, HDC,HIST1H4B,HIST1H4J,PCNA,PLXND1,RBBP7,SOCS3,VIM

CA4 enzyme Activated ANK1,CA1,HEMGN,KEL,RHCE/RHD,SLC4A1,SPTB

SP3 transcriptio

n regulator

ADD3,Ccl2,CDC25B,F2R,FOS,IGF2,IL1A,KLF1,LPL,PTTG1,SERPINH1,SPARC,TGF BR3,TIMP1,VIM

IL1R1 transmemb rane receptor

Ccl2,CXCL10,CXCL2,CXCL3,FOS,IL18,IL1A,LIFR,TIMP1

CDKN2A transcriptio

n regulator

A2M,Ccl2,CCNA2,CCNE1,CDC25B,CXCL10,EHD3,FOS,IL1A,MCM4,MKI67,PCNA, PLAGL1,PLK1,RBBP7,SKP2,VIM

NFE2L2 3.61 transcriptio n regulator

ALAS2,ALDOA,Ccl2,CXCL10,CXCL2,CXCL3,EMCN,GSTA5,GSTP1,HMOX1,IL1A, LPL,Mt1,PSAT1,RAMP2,RBBP7,RELN,SLC2A1,SOCS3,VCAM1

EGF growth

factor

AFP,CAV1,Ccl2,CCND2,CCNE1,DCN,FOS,GSTP1,HMOX1,IGF2,IGFBP2,PCNA,PLA GL1,PTTG1,S100A10,S100A11,SOCS3,SPARC,TIMP1,TIMP3,VCAM1,VIM

DYSF other ANXA2,C1QB,CD48,Cd52,CD55,CXCL10,LCP1,LGALS3,TCEAL9,TIMP1

PI3K (complex) complex Inhibited AQP7,Ccl2,CCND2,CCNE1,CD55,CXCL10,FABP5,FOS,GSTA5,GSTP1,H19,HMOX1,I GF2,IGFBP2,SOCS3,UGCG,VCAM1

IFNG cytokine Inhibited A2M,C1QB,CAV1,Ccl2,CCNA2,CCND2,CD55,CXCL10,CXCL2,CXCL3,EDNRB,EGL N3,F2R,FABP5,FCER1G,FOS,HMOX1,IFITM2,IL18,IL1A,LGALS3,LIFR,LPL,Mt1,PH GDH,PTN,RBBP7,S100A10,SERPINH1,SLC2A1,SLC7A5,SOCS3,TGFBR3,TIMP1,TI MP3,VCAM1

Immunoglobulin complex ALAS2,Ccl2,CCND2,CCNE1,CXCL10,CXCL2,CXCL3,DPYSL2,FCER1G,FOS,HMOX 1,IL1A,SLC25A37,TIMP1,VCAM1

PDGF BB complex Inhibited ADD3,Ccl2,CCNE1,CXCL2,DAB2,DCN,EDNRB,FLNA,FOS,H19,HMOX1,IGF2,LGA LS3,Mt1,PCNA,SOCS3,TIMP1,VCAM1

CD38 enzyme Inhibited ALDOA,ANXA2,CCND2,CCNE1,EGLN3,LGALS3,NDRG1,PSAT1,SLC2A1,SLC7A5, SOCS3,VCAM1,VIM

TICAM1 other Inhibited Ccl2,CXCL10,CXCL2,CXCL3,EDNRB,IL18,IL1A,MCM2,MKI67,SOCS3,TFEC,VCAM 1

LCN2 transporter Inhibited BMP2,Ccl2,CXCL10,CXCL2,CXCL3,HMOX1,IL1A,TAGLN2,VIM

HIPK2 kinase ALAS2,ANK1,CCND2,KLF1,LGALS3,SLC25A37,SLC4A1,SPTB,VIM

Ap1 complex CCNA2,FOS,GSTA5,GSTP1,HBB,HMOX1,IL1A,LPL,NDRG1,SPARC,TIMP1,VCAM1

LDL complex Inhibited BMP2,Ccl2,CDH5,CXCL10,CXCL2,EDNRB,EMB,FOS,HMOX1,IGFBP2,IL1A,MKI67, SOCS3,TGFBR3,VCAM1

IL5 cytokine Inhibited A2M,ALDOA,ANXA2,CCND2,CCNE1,CD55,EGLN3,LUM,NDRG1,PMP22,PSAT1,R BM3,SLC2A1,SLC7A5,SNTB1,VIM

CSF2 cytokine Inhibited Ccl2,CCNA2,CXCL10,CXCL2,F2R,FOS,HDC,IL1A,KLF1,LCP1,MCM6,MKI67,PHGD H,PLK1,PMP22,RBM3,SKA3,SNTB1,SOCS3,TPX2

PTPRJ 3.13 phosphatas

e

Inhibited CCNA2,CXCL2,CXCL3,FOS,HDC,IL18,IL1A,PLAGL1

IKBKG kinase Inhibited BMP2,Ccl2,CXCL2,CXCL3,DCN,FOS,IL1A,LIFR,Mt1,OGN,SOCS3

ERBB2 kinase Inhibited ANXA2,CCNA2,CCND2,CCNE1,CXCL10,CXCL3,EMP1,F2R,FOS,H19,IGF2,IL1A,LG ALS3,LUM,MKI67,NDRG1,PCNA,SKP2,SLC2A1,SPARC,TCEAL9,TIMP3,TUBA1A, VIM

SMAD7 transcriptio n regulator

BGN,BMP2,Ccl2,CCNA2,CCNE1,CXCL10,DCN,HMOX1,PCNA,TIMP1,TIMP3

SRC kinase CA2,CAV1,CCND2,CCNE1,CXCL10,F2R,FOS,HMOX1,PLK1,VCAM1,VIM

DICER1 enzyme AFP,CCND2,FOS,H19,IGF2,IGF2BP1,IGF2BP2,KLF1,LCP1,PMP22,SOCS3,SPARC,VI M

TNFSF11 cytokine Inhibited CA2,CAV1,Ccl2,CCNE1,CXCL3,DAB2,FOS,GRB10,HMOX1,IL1A,LDB2,PLK1,SLC2 A1,SOCS3,VCAM1

IL10 cytokine BMP2,Ccl2,CCND2,CD55,CXCL10,CXCL2,CXCL3,DCN,FCER1G,FOS,HMOX1,IL18,

IL1A,PHGDH,SOCS3,TIMP1,VCAM1

PTGER2 g-protein

coupled receptor

CCNA2,CFP,HDC,HIST1H2AB,IL1A,MKI67,PLK1,TIMP1,TIMP3,TPX2

KCNK9 ion

channel

A2M,CA1,HEMGN,KEL,RHAG,RHCE/RHD,SPTA1

AR ligand-

dependent nuclear receptor

CAV1,CCNA2,CDC25B,EDNRB,EHD3,EMB,FABP5,GPR182,GSN,GSTP1,IGF2,MCM 2,MCM4,NDRG1,PLK1,SKP2,STEAP2,TPX2,VIM

IL1 group Inhibited ADAMTS1,BMP2,Ccl2,CD55,CXCL10,CXCL3,DCN,FOS,H19,HMOX1,SLC2A1,SOCS 3,SPARC,TIMP1,UGCG,VCAM1

ERK group Inhibited BGN,CAV1,Ccl2,CCNE1,CXCL10,CXCL2,DPYSL2,FOS,HMOX1,NDRG1,SLC2A1,TI MP1,TUBA1A,UGCG

GATA1 transcriptio

n regulator

ALAS2,ANK1,CA1,CA2,CCND2,CPA3,HBB,HBG2,KLF1,Podxl,SLC4A1,SPTA1,SPT B

SMARCB1 transcriptio

n regulator

A2M,ADD3,CCNA2,CCNE1,FOS,GSN,IGFBP2,MCM2,MCM4,PTN,SKP2,SPARC

LEP growth

factor

Inhibited AQP7,CAV1,Ccl2,CCNA2,CXCL10,DLK1,ELOVL6,FOS,IGFBP2,LIFR,LPL,PCNA,SO CS3,SPARC,TIMP1,TIMP3,UCP2,VCAM1,VIM

IL1A -4.49 cytokine Inhibited ADAMTS1,CA2,Ccl2,CXCL10,CXCL2,CXCL3,FOS,HDC,HMOX1,IL18,IL1A,SPARC, VCAM1

ADIPOQ other BMP2,CXCL10,CXCL3,DLK1,FOS,HMOX1,LPL,PCNA,TIMP1,UCP2,VCAM1

RELA transcriptio

n regulator

Inhibited A2M,AFP,ARHGDIB,BMP2,CAV1,Ccl2,CXCL10,CXCL2,CXCL3,FOS,HMOX1,IGFB P2,IL1A,LUM,PLK1,VCAM1,VIM

ERK1/2 group Inhibited BMP2,CAV1,Ccl2,CCND2,CXCL10,CXCL3,EMCN,FOS,H19,IL1A,PCNA,PTN,SOCS3 ,TIMP1,VCAM1

MTPN transcriptio

n regulator

Inhibited Ccl2,CCNA2,CCND2,FOS,Mt1,S100A10,SPARC,TUBA1A,VCAM1

CSF1R kinase Inhibited CCND2,CCNE1,FOS,IL1A,PCNA,VCAM1

CSF1 cytokine Inhibited Ccl2,CCND2,CCNE1,CXCL2,CXCL3,F2R,FCER1G,FOS,IL18,IL1A,PCNA,VCAM1

ESR1 6.61 ligand- dependent

nuclear receptor

Inhibited ADD3,BMP2,CA2,CAV1,CCNA2,CCNE1,CD55,CLEC1B,CXCL3,DAB2,FLNA,FOS,F XYD6,GSN,GSTA5,H19,HPGDS,IFITM2,IGF2,IGFBP2,IL1A,KLF1,KLHL13,KNL1,LP L,MKI67,PCNA,PSAT1,PTTG1,SGO2,SKP2,SLC25A4,SLC7A5,VIM

Histone h4 group CCNE1,CXCL10,CXCL3,FOS,GSTP1,IL1A,MCM4,Mt1,PCNA,SOCS3,VCAM1

SOX4 transcriptio

n regulator

ALDH1B1,EMB,EMP1,FCER1G,FOS,Ifitm1,IGF2,Mt1,PPIC,Tpm4,TUBA1A,VIM ACOX1 4.66 enzyme Activated ACER2,ADAMTS1,ANXA2,GSTP1,IGFBP2,LGALS3,LPL,RBM3,TAGLN2,UCP2,UG

CG

TLR4 transmemb

rane receptor

Inhibited BMP2,Ccl2,CCND2,CXCL10,CXCL2,CXCL3,DAB2,DLK1,HDC,HMOX1,IL18,IL1A,P LAGL1,SOCS3,UGCG,VCAM1

SMAD4 transcriptio

n regulator

AFP,BGN,BMP2,Ccl2,CCND2,CCNE1,CDH5,FOS,HMOX1,SLC25A4,TIMP1,TIMP3,V IM

IL6R transmemb

rane receptor

A2M,CXCL10,CXCL2,CXCL3,IGF2,SOCS3,TIMP1,VCAM1

GATA2 transcriptio

n regulator

ALAS2,CDH5,CPA3,EMCN,HDC,HEMGN,KEL,KLF1,Mcpt1,RHAG,RHCE/RHD,SKP 2,SLC4A1,VCAM1

RBL1 transcriptio

n regulator

Activated CCNA2,CCNE1,FOS,MCM2,MCM6,PCNA,PLK1,SKP2

KIT transmemb

rane receptor

Ccl2,CCND2,CPA3,CXCL3,HDC,HMOX1,LGALS3,SOCS3,SPTA1

VEGFA growth

factor

Inhibited ADAMTS1,CAV1,Ccl2,CCNE1,CD55,CDH5,CXCL10,FOS,GRB10,HMOX1,PCNA,RA SGRP3,SPARC,VCAM1

NOD2 other Inhibited BMP2,CXCL10,CXCL2,CXCL3,IL18,IL1A,RASGRP3,SOCS3

IL11 cytokine A2M,ANXA2,DLK1,FOS,SOCS3,TIMP1,VCAM1

NR3C1 ligand-

dependent nuclear receptor

A2M,BMP2,CAV1,Ccl2,CXCL10,CXCL2,CXCL3,DPP7,EMP1,F2R,FCER1G,FOS,GST P1,IL18,IL1A,Mt1,Mt1m/Mt2A,PLAGL1,PRKAR1B,STOM,TIMP3,UGCG,VCAM1

PPARD ligand-

dependent nuclear receptor

AQP7,C1QB,Ccl2,CCND2,CCNE1,GSTA5,IGFBP2,LDHB,LPL,Mcpt1,PCNA,UCP2

STAT1 transcriptio

n regulator

Inhibited A2M,ALAS2,Ccl2,CCND2,CCNE1,CXCL10,CXCL3,EGLN3,FCER1G,FOS,IFITM2,PT N,S100A10,SOCS3

SNAI1 transcriptio CCND2,CCNE1,CD55,CDC25B,CDH5,FLNA,FOS,GSN,SPARC

n regulator

BTK kinase CCND2,CCNE1,CXCL10,CXCL3,EMP1,FABP5,HMOX1,IL18,IL1A

FGFR2 kinase Inhibited AFP,CA2,CCND2,DAB2,GRB10,IGF2,IL1A,LGALS2,TFEC,VCAM1 KLF1 -4.05 transcriptio

n regulator

ALAS2,CD55,HBB,HBG2,SERPINH1,SPTB

PRL cytokine Inhibited A2M,ANXA2,CAV1,CXCL10,DCN,FOS,GPNMB,IGF2,LYVE1,PCNA,SOCS3,SPARC, TIMP1,VIM

VHL transcriptio

n regulator

CA12,CAV1,DAB2,EGLN3,HMOX1,PCNA,SKP2,SLC2A1,SPARC,VIM

PTEN phosphatas

e

CA12,CA2,Ccl2,CCNE1,CDH5,CXCL10,CXCL2,FOS,IGF2,IGFBP2,LGALS3,MKI67,N DRG1,PLK1,PTN,SKP2,SOCS3,VCAM1

CYP1B1 enzyme Inhibited CBX3,CCNE1,HMOX1,IGFBP2,MCM4,Mt1,SKP2

FAS transmemb

rane receptor

ANXA2,BGN,Ccl2,CD48,CXCL10,CXCL2,CXCL3,FOS,GPNMB,IL18,IL1A,LGALS3, LUM,TAGLN2,UGCG,VCAM1

STAT3 transcriptio

n regulator

Inhibited A2M,ALAS2,CCND2,CCNE1,CDH5,CXCL10,CXCL2,CXCL3,FCER1G,FOS,HMOX1,I FITM2,Mt1,NDRG1,PTN,SLC2A1,SOCS3,TIMP1,VIM

APOE transporter BGN,CAV1,Ccl2,CCND2,CXCL3,F2R,FOS,HMOX1,IL1A,LPL,SOCS3,TIMP1,VCAM 1

MITF transcriptio

n regulator

Inhibited APOLD1,CDC25B,EDNRB,FOS,GPNMB,HPGDS,LGALS3,MCM2,MCM4,MCM6,PL K1,TMCC2,TPX2

KRAS enzyme ALDOA,BGN,CAV1,CXCL10,FOS,GPC3,GSN,IFITM2,IGF2,IGF2BP2,IGFBP2,ITM2A

,PLAGL1,SPARC,STOM,VIM RARRES2 15.87 transmemb

rane receptor

Ccl2,CCNA2,CCND2,CD55,CXCL2

PRKCA kinase ARHGDIB,CAV1,CCNE1,CD55,CXCL2,CXCL3,FOS,LPL,VCAM1

ANK1 -3.02 other ANK1,RHAG,RHCE/RHD

CTGF growth

factor

ADAMTS1,AFP,DCN,EGLN3,IGF2,RAMP2,SPARC,TIMP1,TIMP3

AKT1 kinase Inhibited BMP2,CCND2,CCNE1,CXCL10,FABP5,FOS,GSTA5,HMOX1,IGF2,SLC2A1,TGFBR3, TIMP1,VIM

HMOX1 -3.04 enzyme Activated Ccl2,CXCL10,CXCL2,CXCL3,FOS,HMOX1,RELN,SPARC,VCAM1

IGF2 -69.40 growth

factor

BMP2,Ccl2,H19,IFITM2,IGF2,IGFBP2,MCM2,MCM4,NDRG1,OGN,SOCS3

TGFA growth

factor

CXCL10,CXCL2,FOS,GSTP1,PLAGL1,PTTG1,S100A10,VIM

MIF cytokine Inhibited Ccl2,CXCL2,CXCL3,F2R,FOS,RAMP2,TIMP1,VCAM1

BET group ALAS2,HMOX1,KLF1,SLC4A1

C8 complex Ccl2,CXCL2,CXCL3,VCAM1

C9 10.95 other Ccl2,CXCL2,CXCL3,VCAM1

C7 other Ccl2,CXCL2,CXCL3,VCAM1

C3 peptidase Ccl2,CD55,CXCL10,CXCL2,CXCL3,IL1A,UCP2

INSIG1 other CXCL10,CXCL2,CXCL3,DLK1,ELOVL6,FABP5,LPL,STEAP2,UCP2

AMPK complex BMP2,Ccl2,CCND2,CXCL10,HMOX1,LDHB,SLC2A1,UCP2,VIM

WNT5A cytokine ARHGDIB,CXCL2,DAB2,FLNA,IL1A,LCP1,SOCS3,SPARC,VIM

F2R -6.85 g-protein

coupled receptor

Inhibited Ccl2,CD55,CXCL3,F2R,FOS,HMOX1,VCAM1

FAM3B cytokine CAV1,DCN,PTN,RNASE1,SPARC

ERBB3 kinase BGN,CCND2,HMOX1,IGF2,PLK1,SOCS3,SPARC,TIMP3

TAC1 other Inhibited Ccl2,CXCL10,CXCL3,FOS,HDC,HMOX1,IL1A,LDB2

SOCS1 other Activated A2M,Ccl2,CCNE1,CXCL10,CXCL2,FCER1G,FOS,SOCS3,VCAM1

E2F1 transcriptio

n regulator

CA2,CAV1,CCNA2,CCND2,CCNE1,CDC25B,FOS,H19,HIST1H2AB,KIAA0101,MCM 2,MCM4,MCM6,PCNA,PSAT1,VCAM1,VIM

YY1 transcriptio

n regulator

CBX3,CCNA2,FOS,GPC3,HMOX1,MCM4,MCM6,MKI67,PCNA,PLAGL1,PLK1,SLC2 5A4,TNNI1

F2 peptidase Inhibited ALDH1B1,CCNA2,CCND2,CD55,CXCL3,EDNRB,F2R,FOS,HMOX1,RHOJ,SKP2,TA GLN2,VCAM1

RASSF1 other CAV1,CCNA2,CCND2,DAB2,EMP1,FOS,GSN,LDB2

Shc group CCND2,CCNE1,FOS,LPL

S100A8 other A2M,ADAMTS1,C1QB,Ccl2,CXCL10,CXCL2,CXCL3,H19,HMOX1,IL1A,VCAM1

KLF2 transcriptio

n regulator

Ccl2,CD55,CXCL2,HBB,HBG2,IGF2,NDRG1,SLC2A1,TIMP1,VCAM1

E2F4 transcriptio

n regulator

CCNA2,CCNE1,HIST1H2AB,KIAA0101,MCM4,MCM6,MKI67,PCNA,PLK1,PSAT1,P TTG1,TPX2

KLF6 transcriptio

n regulator

Ccl2,CXCL2,DLK1,IL1A,MKI67,PCNA,SERPINH1

IL10RA transmemb

rane receptor

ADD3,BMP2,CA2,DCN,EDNRB,FABP5,IL1A,LUM,OGN,PMP22,SLC2A1,SOCS3,SP ARC,TFEC

JAK2 kinase Inhibited ACER2,Ccl2,CCND2,CXCL10,FOS,Ifitm1,NDN,SOCS3,SPTB

MET kinase Inhibited CCND2,DAB2,FOS,HDC,HMOX1,IL18,PLK1,SOCS3

BDNF growth

factor

ANXA2,BMP2,CCND2,ELOVL6,FLNA,FOS,PCNA,PRKAR1B,RELN,S100A10,SERPI NH1,SPARC,TUBA1A,VIM

Dalam dokumen Supplemental Materials and Methods (Halaman 120-200)

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